Nonsteroidal selective androgen receptor modulators (SARMs): dissociating the anabolic and androgenic activities of the androgen receptor for therapeutic benefit

J Med Chem. 2009 Jun 25;52(12):3597-617. doi: 10.1021/jm900280m.
No abstract available

Publication types

  • Review

MeSH terms

  • Amides / chemistry
  • Amides / pharmacology*
  • Anabolic Agents / chemistry
  • Anabolic Agents / pharmacology*
  • Androgen Receptor Antagonists
  • Androgens / chemistry
  • Androgens / pharmacology*
  • Animals
  • Humans
  • Models, Molecular
  • Quinolones / chemistry
  • Quinolones / pharmacology*
  • Receptors, Androgen / metabolism*
  • Structure-Activity Relationship

Substances

  • Amides
  • Anabolic Agents
  • Androgen Receptor Antagonists
  • Androgens
  • Quinolones
  • Receptors, Androgen
  • propionamide